Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

AZ3451

AZ3451 is a potent protease-activated receptor-2 (PAR2) antagonist with IC50 of 23 nM.

Product Specifications

CAS Number

2100284-59-9

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Protease Activated Receptor (PAR)

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/AZ3451.html

Concentration

10mM

Purity

99.84

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

O=C(C1=CC=C2C(N=C(C3=C(Br)C=C(OCO4)C4=C3)N2[C@H](C5CCCCC5)C)=C1)NC6=CC=C(C#N)C=C6

Molecular Formula

C30H27BrN4O3

Molecular Weight

571.46

Precautions

H302, H315, H319, H335

References & Citations

[1]Cheng RKY, et al. Structural insight into allosteric modulation of protease-activated receptor 2. Nature. 2017 May 4;545 (7652) :112-115.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

PAR2

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Diphenyliodonium Chloride
TRC-D493200-500MG 500 mg

Diphenyliodonium Chloride

Sign In for Pricing
View Details
Mouse Mcm3 activation kit by CRISPRa
GA202603 1 Kit

Mouse Mcm3 activation kit by CRISPRa

Sign In for Pricing
View Details
Frozen Tissue Sections, Rectum
CS629202 5x 5 µm

Frozen Tissue Sections, Rectum

Sign In for Pricing
View Details
GBE1 Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI4E6]
TA500779AM 100 µL

GBE1 Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI4E6]

Sign In for Pricing
View Details
3-Hydroxy Midostaurin
TRC-H939985-2.5MG 2.5 mg

3-Hydroxy Midostaurin

Sign In for Pricing
View Details
Nucleolin (NCL) Goat Polyclonal Antibody
AB0291-100 100 µg

Nucleolin (NCL) Goat Polyclonal Antibody

Sign In for Pricing
View Details