Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

EBI-2511

EBI-2511 is a highly potent and orally active EZH2 inhibitor, with an IC50 of 6 nM in Pfeffiera cell lines, respectively.

Product Specifications

CAS Number

2098546-05-3

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Histone Methyltransferase

Type

Reference compound

Related Pathways

Epigenetics

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/EBI-2511.html

Purity

99.81

Solubility

DMSO : 5 mg/mL (ultrasonic)

Smiles

CCC1=C(C(NCC2=C(C)C=C(C)NC2=O)=O)C(C=C(C3CCN(C(C)C)CC3)O4)=C4C=C1N(C5CCOCC5)CC

Molecular Formula

C34H48N4O4

Molecular Weight

576.77

Precautions

H302, H315, H319, H335

References & Citations

[1]Lu B, et al. Discovery of EBI-2511: A Highly Potent and Orally Active EZH2 Inhibitor for the Treatment of Non-Hodgkin's Lymphoma. ACS Med Chem Lett. 2018 Jan 29;9 (2) :98-102.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

EZH2

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Ube1L (UBA7) Mouse Monoclonal Antibody [Clone ID: OTI2B6]
CF811855 100 µg

Ube1L (UBA7) Mouse Monoclonal Antibody [Clone ID: OTI2B6]

Sign In for Pricing
View Details
Fmoc-Cys (StBu) TentaGel® S AC Resin
SA1109.25G 25 g

Fmoc-Cys (StBu) TentaGel® S AC Resin

Sign In for Pricing
View Details
IGSF5 Human Gene Knockout Kit (CRISPR)
KN420223 1 Kit

IGSF5 Human Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details
KLF5 Rabbit Polyclonal Antibody
AP17518PU-N 400 µL

KLF5 Rabbit Polyclonal Antibody

Sign In for Pricing
View Details
Mouse Interferon alpha 1 Recombinant Rabbit monoclonal Antibody
HA723672 100 µL

Mouse Interferon alpha 1 Recombinant Rabbit monoclonal Antibody

Sign In for Pricing
View Details
4-Chlorophenothiazine
TRC-C374985-1G 1 g

4-Chlorophenothiazine

Sign In for Pricing
View Details