BET-IN-25
BET-IN-25 (compound 7) is an oral bioactive inhibitor of bromodomain (BD1) and BD2, with the IC50s of 0.18 μM and 9.2 μM, respectively[1].
Product Specifications
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/bet-in-25.html
Smiles
CN1C=C(C2=NN(C)C=C2)C(OC(CN3CCN(S(=O)(C)=O)C[C@H]3C)=C4)=C4C1=O
Molecular Formula
C19H25N5O4S
Molecular Weight
419.50
References & Citations
[1]Shuichi Hagihara, et al. Discovery of a potent, orally available furopyridine derivative as a novel selective bromodomain and extra-terminal domain (BET) -first bromodomain (BD1) inhibitor. Bioorg Med Chem Lett. 2024 Sep 1:109:129848.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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