5-HT6R antagonist 4
5-HT6R antagonist 4 (compound 30) is a neutral antagonist of 5-HT6R, with the Ki of 1 nM[1].
Product Specifications
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/5-ht6r-antagonist-4.html
Smiles
FC1=CC(C2=CC=CN2S(=O)(C3=CC(N4CCNCC4)=CC=C3)=O)=CC=C1
Molecular Formula
C20H20FN3O2S
Molecular Weight
385.46
References & Citations
[1]Marcin Drop, et al. 5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives. Eur J Med Chem. 2024 Sep 5:275:116615.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT6 Receptor
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