PROTAC BET-binding moiety 2
PROTAC BET-binding moiety 2 is an inhibitor of BET bromodomain[1].
Product Specifications
CAS Number
916493-82-8
UNSPSC
12352005
Hazard Statement
H315, H319, H335
Target
Ligands for Target Protein for PROTAC
Type
Reference compound
Related Pathways
PROTAC
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/PROTAC_BET-binding_moiety_2.html
Purity
99.77
Solubility
DMSO : 42.86 mg/mL (ultrasonic)
Smiles
CC1=C(C(O)=O)SC2=C1C(C3=CC=C(Cl)C=C3)=N[C@@H](CC(OC)=O)C4=NN=C(C)N24
Molecular Formula
C20H17ClN4O4S
Molecular Weight
444.89
Precautions
H315, H319, H335
References & Citations
[1]James E. Bradner, et al. Bivalent bromodomain inhibtors and uses thereof. WO2017091673A2.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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