CAY10471 (Racemate)
CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM) . CAY10471 Racemate also has effect on mouse and rat orthologs of CRTH2[1].
Product Specifications
CAS Number
844639-57-2
Product Name Alternative
TM30089 (Racemate)
UNSPSC
12352005
Hazard Statement
H315, H317, H319, H400, H410
Target
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Cancer-programmed cell death
Field of Research
Cancer; Endocrinology
Assay Protocol
https://www.medchemexpress.com/CAY10471_Racemate.html
Concentration
10mM
Purity
99.00
Solubility
DMSO : 150 mg/mL (ultrasonic)
Smiles
O=C(O)CN1C2=C(C3=C1C=CC=C3)CC(N(S(=O)(C4=CC=C(F)C=C4)=O)C)CC2
Molecular Formula
C21H21FN2O4S
Molecular Weight
416.47
Precautions
H315, H317, H319, H400, H410
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DP
Available Sizes
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog
