GPR4 antagonist 1
GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.
Product Specifications
CAS Number
[1197879-16-5]
UNSPSC
12352005
Target
GPR4
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cancer
Assay Protocol
https://www.medchemexpress.com/GPR4_antagonist_1.html
Purity
98.92
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
CC1=C2C(N(CC3=CC=C(/C=C/CN4CCN(C(C)C)CC4)C=C3)C(CC)=N2)=NC(C)=C1
Molecular Formula
C27H37N5
Molecular Weight
431.62
References & Citations
[1]ARYL SULFONOHYDRAZIDES. US 20090291942 A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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