GPR4 antagonist 1

GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.

Product Specifications

CAS Number

[1197879-16-5]

UNSPSC

12352005

Target

GPR4

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology; Cancer

Assay Protocol

https://www.medchemexpress.com/GPR4_antagonist_1.html

Purity

98.92

Solubility

DMSO : 125 mg/mL (ultrasonic)

Smiles

CC1=C2C(N(CC3=CC=C(/C=C/CN4CCN(C(C)C)CC4)C=C3)C(CC)=N2)=NC(C)=C1

Molecular Formula

C27H37N5

Molecular Weight

431.62

References & Citations

[1]ARYL SULFONOHYDRAZIDES. US 20090291942 A1.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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