UFP-512
UFP-512 is a selective and potent σ-opioid receptor (DOP receptor) peptidic agonist with antidepressant- and anxiolytic-like effects. UFP-512 exhibits as a potent agonist on adenylyl cyclase inhibition and Erk1/2 activation. UFP-512 induces phosphorylation of DOP receptors on Ser363 with a low desensitization of the cAMP pathway. UFP-512 is promising for research of mood disorders[1].
Product Specifications
CAS Number
480446-44-4
UNSPSC
12352005
Target
Adenylate Cyclase; ERK; Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; MAPK/ERK Pathway; Neuronal Signaling; Stem Cell/Wnt
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ufp-512.html
Smiles
CC(C=C(C=C1C)O)=C1C[C@H](N)C(N2[C@@H](CC3=CC=CC=C3C2)C(N[C@H](C4=NC5=CC=CC=C5N4)CC(O)=O)=O)=O
Molecular Formula
C31H33N5O5
Molecular Weight
555.62
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog
Recombinant Salmonella schwarzengrund NADH-quinone oxidoreductase subunit B (nuoB)
Recombinant Salmonella schwarzengrund NADH-quinone oxidoreductase subunit B (nuoB)
Recombinant Salmonella schwarzengrund NADH-quinone oxidoreductase subunit B (nuoB)
Recombinant Salmonella schwarzengrund NADH-quinone oxidoreductase subunit B (nuoB)
Recombinant Salmonella schwarzengrund NADH-quinone oxidoreductase subunit B (nuoB)