Bay 59-3074

Bay 59-3074 is a selective cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively. Bay 59-3074 has analgesic properties[1].

Product Specifications

CAS Number

[406205-74-1]

UNSPSC

12352005

Hazard Statement

H302, H315, H320, H335

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/Bay-59-3074.html

Purity

98.60

Solubility

DMSO : ≥ 100 mg/mL

Smiles

O=S(CCCC(F)(F)F)(OC1=CC=CC(OC2=CC=CC(C(F)(F)F)=C2C#N)=C1)=O

Molecular Formula

C18H13F6NO4S

Molecular Weight

453.36

Precautions

H302, H315, H320, H335

References & Citations

[1]De Vry J et al. 3-[2-cyano-3- (trifluoromethyl) phenoxy]phenyl-4,4,4-trifluoro-1-butanesulfonate (BAY 59-3074) : a novelcannabinoid Cb1/Cb2 receptor partial agonist with antihyperalgesic and antiallodynic effects. J Pharmacol Exp Ther. 2004 Aug;310 (2) :620-32.