AC-7954 (free base)
AC-7954 free base is a selective nonpeptidic urotensin receptor agonist (EC50: 300 nM at the human UII receptor) [1].
Product Specifications
CAS Number
734528-95-1
UNSPSC
12352005
Target
Urotensin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/ac-7954-free-base.html
Smiles
O=C1OC(CC2=C1C=CC=C2)(CCN(C)C)C3=CC=C(C=C3)Cl
Molecular Formula
C19H20ClNO2
Molecular Weight
329.82
References & Citations
[1]Croston GE, et al. Discovery of the first nonpeptide agonist of the GPR14/urotensin-II receptor: 3- (4-chlorophenyl) -3- (2- (dimethylamino) ethyl) isochroman-1-one (AC-7954) . J Med Chem. 2002 Nov 7;45 (23) :4950-3.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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