(N-Me-Tyr1, N-Me-Arg7, D-Leu-NHEt8) -Dynorphin A (1-8)
Selected Variant
HY-P4679
Size: 1 Each
(N-Me-Tyr1, N-Me-Arg7, D-Leu-NHEt8) -Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) analog, is a kappa opioid receptor (KOR) agonist[1].
Product Specifications
CAS Number
103613-84-9
Product Name Alternative
E2078
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/n-me-tyr1-n-me-arg7-d-leu-nhet8-dynorphin-a-1-8.html
Solubility
H2O
Smiles
CCNC([C@@H](CC(C)C)NC([C@H](CCCNC(N)=N)N(C)C([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](NC(CNC(CNC([C@@H](NC)CC1=CC=C(C=C1)O)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O
Molecular Formula
C50H81N15O9
Molecular Weight
1036.27
References & Citations
[1]Butelman ER, et al. Effects of E-2078, a stable dynorphin A (1-8) analog, on sedation and serum prolactin levels in rhesus monkeys. Psychopharmacology (Berl) . 1999 Nov;147 (1) :73-80.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
Phase 2
Isoform
κ Opioid Receptor/KOR
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