(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
Product Specifications
UNSPSC Description
(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) (HY-P2159) analog, is a kappa opioid receptor (KOR) agonist[1].
Target Antigen
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/n-me-tyr1-n-me-arg7-d-leu-nhet8-dynorphin-a-1-8.html
Solubility
H2O
Smiles
CCNC([C@@H](CC(C)C)NC([C@H](CCCNC(N)=N)N(C)C([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](NC(CNC(CNC([C@@H](NC)CC1=CC=C(C=C1)O)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O
Molecular Weight
1036.27
References & Citations
[1]Butelman ER, et al. Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys. Psychopharmacology (Berl). 1999 Nov;147(1):73-80.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-P4679/N-Me-Tyr1-N-Me-Arg7-D-Leu-NHEt8-Dynorphin-A-1-8-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-P4679/
Clinical Information
Phase 2
CAS Number
103613-84-9
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
MBS2906332-03 5x 96 Well
Chicken FUNDC1 / FUN14 domain-containing protein 1 ELISA Kit
Ask
View Details 
MBS2906332-04 10x 96 Well
Chicken FUNDC1 / FUN14 domain-containing protein 1 ELISA Kit
Ask
View Details