(αR,8aS) -GSK1614343
(αR,8aS) -GSK1614343 is the isomer of GSK1614343. GSK1614343 is the potent antagonist of growth hormone secretagogues type 1a (GHS1a) receptors[1].
Product Specifications
CAS Number
1092476-84-0
UNSPSC
12352005
Target
GHSR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/αr-8as-gsk1614343.html
Purity
99.72
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
FC(F)(F)C1=CC(C(F)(F)F)=CC(NNC([C@@H](C2=CN=CC=C2)N3C[C@@]4([H])N(CCC4)CC3)=O)=C1
Molecular Formula
C22H23F6N5O
Molecular Weight
487.44
References & Citations
[1]Perdonà E, et al. Pharmacological characterization of the ghrelin receptor antagonist, GSK1614343 in rat RC-4B/C cells natively expressing GHS type 1a receptors. Eur J Pharmacol. 2011;650 (1) :178-183.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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