FFAR1/FFAR4 agonist-1
FFAR1/FFAR4 agonist-1 (compound 83) is a FFAR1/FFAR4 agonist with the EC50 of 1 nM A and 4nM for FFAR1 and FFAR4, respectively. FFAR1/FFAR4 agonist-1 can be used for study of glycemic control[1].
Product Specifications
CAS Number
2839486-16-5
UNSPSC
12352005
Target
Free Fatty Acid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Metabolic Disease; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/ffar1-ffar4-agonist-1.html
Smiles
O=C1N(CCC1)C2=CC(OCC3=NC(NCCC4=CC(Cl)=CC=C4Cl)=NC(N)=N3)=CC(C)=C2
Molecular Formula
C23H24Cl2N6O2
Molecular Weight
487.38
References & Citations
[1]Lückmann M, et al. Optimization of First-in-Class Dual-Acting FFAR1/FFAR4 Allosteric Modulators with Novel Mode of Action. ACS Med Chem Lett. 2022;13 (12) :1839-1847. Published 2022 Nov 2.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
![Nuclear Receptor Corepressor Mouse Monoclonal Antibody [A6H12]](https://cdn.genprice.uk/products/992/68dd1c8b061270361ea8145b/imageurl/ha600055.webp)
HA600055 100 µL
Nuclear Receptor Corepressor Mouse Monoclonal Antibody [A6H12]
Sign In for Pricing
View Details 
10-3005-F-25 25 µg
Monoclonal Antibody to TLR8/CD288 FITC Conjugated (Clone: ABM15F6)
Sign In for Pricing
View Details 