C (phg-isoDGR- (NMe) k) (TFA)
C (phg-isoDGR- (NMe) k) TFA is a selective and potent α5β1-integrin ligand with an IC50 of 2.9 nM[1].
Product Specifications
UNSPSC
12352200
Target
Integrin
Type
Biochemical Assay Reagents
Related Pathways
Cytoskeleton
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/c-phg-isod-g-r-nme-k-tfa.html
Purity
99.63
Solubility
DMSO : 250 mg/mL (ultrasonic)
Smiles
O=C(CNC(C[C@@H](C(O)=O)NC([C@@H](C1=CC=CC=C1)NC([C@H]2CCCCN)=O)=O)=O)N[C@@H](CCCNC(N)=N)C(N2C)=O.OC(C(F)(F)F)=O
Molecular Formula
C29H42F3N9O9
Molecular Weight
717.69
References & Citations
[1]Kapp TG, et al. N-Methylation of isoDGR Peptides: Discovery of a Selective α5β1-Integrin Ligand as a Potent Tumor Imaging Agent. J Med Chem. 2018 Mar 22;61 (6) :2490-2499.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, sealed storage, away from moisture)
Scientific Category
Biochemical Assay Reagents
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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