(±) -BAK2-66
(±) -BAK2-66 is a selectivity dopamine D3 receptor antagonist with theKi values of 1nM and 960 nM for D3R and D2R, respectively. (±) -BAK2-66 can be used for study in animal models of addiction[1].
Product Specifications
CAS Number
1301178-83-5
UNSPSC
12352005
Target
Dopamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/racemic-bak2-66.html
Smiles
O=C(NCCC(CN1CCN(CC1)C2=CC=CC(Cl)=C2Cl)F)C3=CC4=CC=CC=C4O3
Molecular Formula
C23H24Cl2FN3O2
Molecular Weight
464.36
References & Citations
[1]Kumar V, et al. Chiral Resolution and Serendipitous Fluorination Reaction for the Selective Dopamine D3 Receptor Antagonist BAK2-66. ACS Med Chem Lett. 2014;5 (6) :647-651. Published 2014 Mar 24.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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