GPR55 agonist 3
GPR55 agonist 3 (Compound 26) is a GPR55 agonist (EC50: 0.239 nM, and 1.76 nM for hGPR55 and rGPR55) . GPR55 agonist 3 induces β-arrestin recruitment to human GPR55 (EC50: 6.2 nM) [1].
Product Specifications
CAS Number
3006105-44-5
UNSPSC
12352005
Target
GPR55
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gpr55-agonist-3.html
Purity
99.17
Solubility
DMSO : 250 mg/mL (ultrasonic)
Smiles
FC(F)(F)CC1=CN=CC(C2=CN=C(N[C@@H](C3=CC=C(F)C=C3)C)C=N2)=C1
Molecular Formula
C19H16F4N4
Molecular Weight
376.35
References & Citations
[1]Hewer RC, et al. Discovery and Characterization of Novel CNS-Penetrant GPR55 Agonists. J Med Chem. 2023 Sep 28;66 (18) :12858-12876.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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