Nerisopam
Nerisopam is an orally active gamma-aminobutyric acid (GABA) receptor agonist. Nerisopam is an anxiolytic and antipsychotic homophthalazine. Nerisopam induces rapid, intense expression of Fos-like immunoreactivity in the rostral, dorsomedial and lateral parts of the striatum in the rat[1].
Product Specifications
CAS Number
[102771-12-0]
Product Name Alternative
GYKI52322; EGIS-6775
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/nerisopam.html
Solubility
10 mM in DMSO
Smiles
NC1=CC=C(C=C1)C2=NN=C(CC3=CC(OC)=C(C=C32)OC)C
Molecular Formula
C18H19N3O2
Molecular Weight
309.36
References & Citations
[1]Palkovits M, et al. Anxiolytic homophthalazines increase Fos-like immunoreactivity in selected brain areas of the rat. Eur J Pharmacol. 1997 Jul 16;331 (1) :53-63.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Available Sizes
Curated Selection
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