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HI-TOPK-032

Product Specifications

UNSPSC Description

HI-TOPK-032 is a potent and specific TOPK inhibitor.

Target Antigen

TOPK

Type

Reference compound

Related Pathways

Cell Cycle/DNA Damage

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/HI-TOPK-032.html

Purity

98.83

Solubility

DMSO : 2.5 mg/mL (ultrasonic;warming;heat to 60°C)

Smiles

O=C(C1=CC=CS1)NC2=CC3=C(C#N)C4=NC5=CC=CC=C5N=C4N3C=C2

Molecular Weight

369.40

References & Citations

[1]Kim DJ, et al. Novel TOPK inhibitor HI-TOPK-032 effectively suppresses colon cancer growth. Cancer Res. 2012 Jun 15;72(12):3060-8.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-101550/HI-TOPK-032-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-101550/HI-TOPK-032-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

487020-03-1

Available Sizes

Curated Selection

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