Y4R agonist-2

Y4R agonist-2 is a Y4R agonist with a Ki of 0.033 nM.

Product Specifications

CAS Number

[2757328-63-3]

UNSPSC

12352209

Target

Neuropeptide Y Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/y4r-agonist-2.html

Solubility

10 mM in DMSO

Smiles

O=C([C@@H](NC(CC1)=O)CCCNC(N)=N)N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CCCNC(N)=N)=O)CC(C)C)=O)CCCNC(NC(NCCCCNC1=O)=O)=N)=O)CC3=CNC4=CC=CC=C34

Molecular Formula

C53H81N19O10

Molecular Weight

1144.33

References & Citations

[1]Konieczny A, et al. N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y4 Receptor Ligands Results in Picomolar Binding Constants. J Med Chem. 2021 Nov 8.