Herkinorin
Product Specifications
UNSPSC Description
Herkinorin is a potent and selective agonist of µ opioid receptor with a Ki of 45 nM Herkinorin is widely used for pain research[1].
Target Antigen
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/herkinorin.html
Solubility
10 mM in DMSO
Smiles
O=C([C@H](C[C@H](OC(C1=CC=CC=C1)=O)C([C@@]23[H])=O)[C@]2(C)CC[C@@]([C@]3(C)C[C@@H](C4=COC=C4)O5)([H])C5=O)OC
Molecular Weight
494.53
References & Citations
[1]Lamb K, et al. Antinociceptive effects of herkinorin, a MOP receptor agonist derived from salvinorin A in the formalin test in rats: new concepts in mu opioid receptor pharmacology: from a symposium on new concepts in mu-opioid pharmacology. Drug Alcohol Depend. 2012 Mar 1;121(3):181-8.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-121415/Herkinorin-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-121415/
Clinical Information
No Development Reported
CAS Number
862073-77-6
Available Sizes
Curated Selection
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