(S, S) -CPI-1612
(S, S) -CPI-1612 is the isomer of CPI-1612 (HY-136285), and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity[1].
Product Specifications
CAS Number
[2374971-82-9]
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
Histone Acetyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/s-s-cpi-1612.html
Purity
99.88
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
CN(N=C1)C=C1C(C=N2)=CC=C2NC([C@H](C3=CC=CC=C3)NC[C@H](C4=CC=C(C=C4)C#N)C)=O
Molecular Formula
C27H26N6O
Molecular Weight
450.53
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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