(S,S)-CPI-1612
Product Specifications
UNSPSC Description
(S,S)-CPI-1612 is the isomer of CPI-1612 (HY-136285), and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity[1].
Target Antigen
Histone Acetyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/s-s-cpi-1612.html
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
CN(N=C1)C=C1C(C=N2)=CC=C2NC([C@H](C3=CC=CC=C3)NC[C@H](C4=CC=C(C=C4)C#N)C)=O
Molecular Weight
450.53
References & Citations
[1]Wang F, et al. Microstructure of poly(gamma-glutamic acid) produced by Bacillus subtilis consisting of clusters of D- and L-glutamic acid repeating units. J Agric Food Chem. 2008 Jun 11;56(11):4225-8.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-145386/S-S-CPI-1612-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-145386/S-S-CPI-1612-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
2374971-82-9
Available Sizes
Curated Selection
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