(R) -VT104
(R) -VT104 is the R-enantiomer of VT104. (R) -VT104 shows an IC50 value of 0.1-1 μΜ for firefly luciferase. VT104 is an orally active and pan-TEAD auto-palmitoylation inhibitor[1].
Product Specifications
CAS Number
[2417718-26-2]
UNSPSC
12352005
Hazard Statement
H315, H319, H335
Target
YAP
Type
Reference compound
Related Pathways
Stem Cell/Wnt
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/r-vt104.html
Purity
99.93
Solubility
DMSO : ≥ 100 mg/mL
Smiles
O=C(C1=CC=C2C(C3=CC=C(C(F)(F)F)C=C3)=CC=CC2=C1)N[C@@H](C4=NC=CC=C4)C
Molecular Formula
C25H19F3N2O
Molecular Weight
420.43
Precautions
H315, H319, H335
References & Citations
[1]Konradi, Andrei W, et al. Preparation of substituted naphthalene-2-carboxamide derivatives useful for treatment of cancer. WO2020097389.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
CXorf48 (CT55) (NM_017863) Human Tagged ORF Clone Lentiviral Particle
