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SY-LB-57

Product Specifications

UNSPSC Description

SY-LB-57 is a highly potent bone morphogenetic protein (BMP) receptor signaling agonist. SY-LB-57 can be used in studies of diseases such as fractures and pulmonary arterial hypertension[1].

Target Antigen

TGF-β Receptor

Type

Reference compound

Related Pathways

TGF-beta/Smad

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease; Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/sy-lb-57.html

Solubility

DMSO : 16.67 mg/mL (ultrasonic;warming;heat to 60°C)

Smiles

COC1=CC2=C(NC(C3=NC4=CC=CC=C4N3)=C2)C=C1

Molecular Weight

263.29

References & Citations

[1]Sheyda Najafi, et al. Discovery of a novel class of benzimidazoles as highly effective agonists of bone morphogenetic protein (BMP) receptor signaling. Sci Rep. 2022 Jul 15;12(1):12146.

Shipping Conditions

Room Temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-150793/SY-LB-57-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-150793/SY-LB-57-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

2253719-35-4

Available Sizes

Curated Selection

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