Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Cariprazine-d6

Cariprazine-d6 is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM) [1].

Product Specifications

CAS Number

1308278-67-2

Product Name Alternative

RGH-188-d6

UNSPSC

12352005

Hazard Statement

H302+H312+H332, H315, H319

Target

5-HT Receptor; Dopamine Receptor

Type

Isotope-Labeled Compounds

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Purity

98.74

Solubility

DMSO : 2mg/mL (ultrasonic; warming; heat to 60°C)

Smiles

O=C(N[C@H]1CC[C@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C([2H])([2H])[2H])C([2H])([2H])[2H]

Molecular Formula

C21H26D6Cl2N4O

Molecular Weight

433.45

Precautions

H302+H312+H332, H315, H319

References & Citations

[1] Seneca N, et al. Occupancy of dopamine D2 and D3 and serotonin 5-HT1A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography. Psychopharmacology (Berl) . 2011 Dec;218 (3) :579-8

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Isotope-Labeled Compounds

Clinical Information

No Development Reported

Isoform

5-HT1 Receptor; mLAG-3

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

(S)-(+)-Pyrethrolone
TRC-P330780-250MG 250 mg

(S)-(+)-Pyrethrolone

Sign In for Pricing
View Details
Tissue FFPE Sections, Lung
CS809239 5x 5 µm

Tissue FFPE Sections, Lung

Sign In for Pricing
View Details
Mitochondrial Marker (MTC754), Biotin conjugate, 0.1mg/mL
BNCB0754-100 1x 100 µL

Mitochondrial Marker (MTC754), Biotin conjugate, 0.1mg/mL

Sign In for Pricing
View Details
Chromogranin A (LK2H10 + PHE5), CF568 conjugate, 0.1mg/mL
BNC680698-100 1x 100 µL

Chromogranin A (LK2H10 + PHE5), CF568 conjugate, 0.1mg/mL

Sign In for Pricing
View Details
Human BTNL10 activation kit by CRISPRa
GA119084 1 Kit

Human BTNL10 activation kit by CRISPRa

Sign In for Pricing
View Details
Recombinant EFEMP1 Antibody
RC-5695-01 50 μL

Recombinant EFEMP1 Antibody

Sign In for Pricing
View Details