CYT-1010
Product Specifications
UNSPSC Description
CYT-1010 is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively[1].
Target Antigen
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cyt-1010.html
Purity
99.74
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
OC1=CC=C(C=C1)C[C@@H](C(N[C@H](CCCCNC2=O)C(N[C@@H](CC3=CNC4=C3C=CC=C4)C(N[C@H]2CC5=CC=CC=C5)=O)=O)=O)N
Molecular Weight
624.73
References & Citations
[1]Theodore E. Maione, Novel therapeutic uses of mu-opiate receptor peptides. WO2013173730A2.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-123534/CYT-1010-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-123534/CYT-1010-SDS-MedChemExpress.pdf
Clinical Information
Phase 1
CAS Number
213769-33-6
Available Sizes
Curated Selection
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