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PROTAC DYRK2 degrader 1

Product Specifications

UNSPSC Description

PROTAC DYRK2 degrader 1 (compound CP134) is a PROTAC degrader of DYRK2 (Red: DYRK2 inhibitor(HY-161598), black: linker (HY-42776), Blue: E3 ligase ligand (HY-10984))[1].

Target Antigen

PROTACs

Type

Reference compound

Related Pathways

PROTAC

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/protac-dyrk2-degrader-1.html

Smiles

O=C(NCCOCCOCCOCCNC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)CN4C/C(C(/C(C4)=C/C5=CC=CC=C5Br)=O)=C\C6=CC=CC=C6Br

Molecular Weight

921.63

References & Citations

[1]Jian Chen, et al.Discovery of the First Potent DYRK2 Proteolysis Targeting Chimera Degraders. ACS Med. Chem. Lett. 2024, 15, 5, 659–666.

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-161597/PROTAC-DYRK2-degrader-1-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-161597/

Clinical Information

No Development Reported

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