DYR530
Product Specifications
CAS Number
2410298-39-2
UNSPSC Description
DYR530 is a ligand for target protein (protein kinases DYRK1A) for PROTAC (HY-168194)[1].
Target Antigen
DYRK; Ligands for Target Protein for PROTAC
Type
Reference compound
Related Pathways
PROTAC;Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/dyr530.html
Smiles
CN1CCN(C2=CC=C(N3C(C)=NC4=CC=C(C5=CC(N)=NC=C5)N=C43)C=C2F)CC1
Molecular Weight
417.48
References & Citations
[1]Wilms G, et, al. Discovery and Functional Characterization of a Potent, Selective, and Metabolically Stable PROTAC of the Protein Kinases DYRK1A and DYRK1B. J Med Chem. 2024 Oct 10;67(19):17259-17289.
Shipping Conditions
Room temperature
Clinical Information
No Development Reported
Frequently Asked Questions
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