ARM1
ARM1 (4BSA) is a potent aminopeptidase and epoxide hydrolase inhibitor. ARM1 shows aminopeptidase inhibitory activity with an IC50 7.61 µM and epoxide hydrolase inhibitory activity with an IC50 12.4 µM[1].
Product Specifications
CAS Number
[68729-05-5]
Product Name Alternative
4BSA
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Aminopeptidase; Epoxide Hydrolase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/arm1.html
Purity
99.60
Solubility
DMSO : 250 mg/mL (ultrasonic)
Smiles
NC1=NC(C(C=C2)=CC=C2CC3=CC=CC=C3)=CS1
Molecular Formula
C16H14N2S
Molecular Weight
266.37
Precautions
H302, H315, H319, H335
References & Citations
[1]El-Naggar MH, et al. Synthesis, docking, cytotoxicity, and LTA4H inhibitory activity of new gingerol derivatives as potential colorectal cancer therapy. Bioorg Med Chem. 2017;25 (3) :1277-1285.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 3
Available Sizes
Curated Selection
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