ARM1

ARM1 (4BSA) is a potent aminopeptidase and epoxide hydrolase inhibitor. ARM1 shows aminopeptidase inhibitory activity with an IC50 7.61 µM and epoxide hydrolase inhibitory activity with an IC50 12.4 µM[1].

Product Specifications

CAS Number

[68729-05-5]

Product Name Alternative

4BSA

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Aminopeptidase; Epoxide Hydrolase

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/arm1.html

Purity

99.60

Solubility

DMSO : 250 mg/mL (ultrasonic)

Smiles

NC1=NC(C(C=C2)=CC=C2CC3=CC=CC=C3)=CS1

Molecular Formula

C16H14N2S

Molecular Weight

266.37

Precautions

H302, H315, H319, H335

References & Citations

[1]El-Naggar MH, et al. Synthesis, docking, cytotoxicity, and LTA4H inhibitory activity of new gingerol derivatives as potential colorectal cancer therapy. Bioorg Med Chem. 2017;25 (3) :1277-1285.