Quinacainol
Quinacainol (PK 10139) is an inhibitor for sodium current with an EC50 of 95 µM. Quinacainol exhibits antiarrhythmic activity by affecting the electrophysiological properties of the heart[1].
Product Specifications
CAS Number
86073-85-0
Product Name Alternative
PK 10139
UNSPSC
12352005
Target
Sodium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/quinacainol.html
Smiles
OC(CCC1CCNCC1)C2=CC(C(C)(C)C)=NC3=CC=CC=C23
Molecular Formula
C21H30N2O
Molecular Weight
326.48
References & Citations
[1]Rougeot C, et al. PK 10139 and quinidine: interactions with digoxin concentrations in rats and dogs[J]. Journal of pharmacy and pharmacology, 1984, 36 (5) : 347-349.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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