(d (CH2) 51, Tyr (Me) 2, Arg8) -Vasopressin

(d (CH2) 51, Tyr (Me) 2, Arg8) -Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist[1].

Product Specifications

CAS Number

[73168-24-8]

Product Name Alternative

SKF 100273

UNSPSC

12352209

Hazard Statement

H332

Target

Vasopressin Receptor

Type

Peptides

Related Pathways

GPCR/G Protein

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/d-ch2-51-tyr-me-2-arg8-vasopressin.html

Solubility

H2O

Smiles

O=C1CC2(CCCCC2)SSC[C@@](NC([C@@H](NC([C@H](CCC(N)=O)NC([C@@](CC3=CC=CC=C3)([H])NC([C@H](CC4=CC=C(OC)C=C4)N1)=O)=O)=O)CC(N)=O)=O)([H])C(N5[C@@H](CCC5)C(N[C@@H](CCCNC(N)=N)C(NCC(N)=O)=O)=O)=O

Molecular Formula

C52H74N14O12S2

Molecular Weight

1151.36

Precautions

H332

References & Citations

[1]Arai Y, et al. New topics in vasopressin receptors and approach to novel drugs: research and development of conivaptan hydrochloride (YM087), a drug for the treatment of hyponatremia. J Pharmacol Sci. 2009 Jan;109 (1) :53-9.