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MGH-CP1

Product Specifications

CAS Number

896657-58-2

Target

TEAD

Applications

Hippo

Smiles

O=C (CSC1=NN=C[NH]1) NC2=CC=C (C=C2) C34CC5CC (CC (C5) C3) C4

Molecular Formula

C20H24N4OS

Additionnal Information

MGH-CP1 is a potent and selective inhibitor of transcriptional enhanced associate domain (TEAD) palmitoylation. MGH-CP1 exhibits dose-dependent and potent inhibition of TEAD2/4 auto-palmitoylation in vitro with IC50 of 710 nM and 672 nM, respectively.

Storage Conditions

4°C, away from moisture and light.

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