GSK046 (iBET-BD2)
Product Specifications
CAS Number
2474876-09-8
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC (OC1=CC (=CC (=C1NC (C) =O) F) C (=O) NC2CCC (O) CC2) C3=CC=CC=C3
Molecular Formula
C23H27FN2O4
Additionnal Information
GSK046 (iBET-BD2) is a selective and orally active inhibitor of BET (bromodomain and extraterminal domain) with IC50 of 264 nM, 98 nM, 49 nM and 214 nM for BRD2BD2, BRD3BD2, BRD4BD2 and BRDTBD2, respectively. GSK046 exhibits immunomodulatory activity.
Storage Conditions
3 years -20°C powder
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