Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

RK-287107

Product Specifications

CAS Number

2171386-10-8

Target

PARP

Applications

DNA Damage/DNA Repair

Smiles

C1CCC2=C (C1) C (=O) NC (=N2) N3CCC4 (CC3) CN (C5=C4C (=CC (=C5) F) F) CCO

Molecular Formula

C22H26F2N4O2

Additionnal Information

RK-287107 is a novel, potent and selective tankyrase inhibitor with antitumor activity. RK-287107 inhibits tankyrase-1 and tankyrase-2 in vitro with IC50 of 14.3 nM and 10.6 nM.

Storage Conditions

3 years -20°C powder

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-01 0.02 mg (E-Coli)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details
Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-02 0.1 mg (E-Coli)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details
Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-03 0.02 mg (Yeast)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details
Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-04 0.1 mg (Yeast)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details
Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-05 0.02 mg (Baculovirus)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details
Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)
MBS1121334-06 0.02 mg (Mammalian-Cell)

Recombinant Escherichia coli O6 Orotate phosphoribosyltransferase (pyrE)

Sign In for Pricing
View Details