Delgocitinib (JTE-052)
Product Specifications
CAS Number
1263774-59-9
Target
JAK
Applications
Angiogenesis
Smiles
CC1CN (C12CCN (C2) C3=NC=NC4=C3C=CN4) C (=O) CC#N
Molecular Formula
C16H18N6O
Additionnal Information
Delgocitinib (JTE-052) is a specific JAK inhibitor with IC50s of 2.8, 2.6, 13 and 58 nM for JAK1, JAK2, JAK3 and Tyk2, respectively.
Storage Conditions
3 years -20°C powder
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