Tinostamustine (EDO-S101)
Product Specifications
CAS Number
1236199-60-2
Target
HDAC
Applications
DNA Damage/DNA Repair
Smiles
CN1C2=C (C=C (C=C2) N (CCCl) CCCl) N=C1CCCCCCC (=O) NO
Molecular Formula
C19H28Cl2N4O2
Additionnal Information
Tinostamustine (EDO-S101) is a first-in-class alkylating deacetylase inhibitor with IC50 values of 9 nM, 9 nM, 25 nM and 107 nM for HDAC1, HDAC2, HDAC3 and HDAC8 (Class 1 HDACs) respectively and 6 nM, 72 nM for HDAC6 and HDAC10 (Class II HDACs) .
Storage Conditions
3 years -20°C powder
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS6208698-01 0.1 mL
SP3 (Sp3 Transcription Factor, DKFZp686O1631, SPR-2) (MaxLight 490)
Sign In for Pricing
View Details MBS6208698-02 5x 0.1 mL
SP3 (Sp3 Transcription Factor, DKFZp686O1631, SPR-2) (MaxLight 490)
Sign In for Pricing
View Details MBS1285966-01 0.05 mg (E-Coli)
Recombinant Chromobacterium violaceum N-acetyl-gamma-glutamyl-phosphate reductase (argC)
Sign In for Pricing
View Details MBS1285966-02 0.05 mg (Yeast)
Recombinant Chromobacterium violaceum N-acetyl-gamma-glutamyl-phosphate reductase (argC)
Sign In for Pricing
View Details MBS1285966-03 0.2 mg (E-Coli)
Recombinant Chromobacterium violaceum N-acetyl-gamma-glutamyl-phosphate reductase (argC)
Sign In for Pricing
View Details MBS1285966-04 0.05 mg (Baculovirus)
Recombinant Chromobacterium violaceum N-acetyl-gamma-glutamyl-phosphate reductase (argC)
Sign In for Pricing
View Details