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A-804598

Product Specifications

CAS Number

1125758-85-1

Target

P2 Receptor

Applications

Neuronal Signaling

Smiles

CC (C1=CC=CC=C1) N=C (NC#N) NC2=CC=CC3=C2C=CC=N3

Molecular Formula

C19H17N5

Additionnal Information

A-804598 is a selective P2X7R antagonist with high affinity at rat (IC50 = 10 nM), mouse (IC50 = 9 nM) and human (IC50 = 11 nM) P2X7 receptors.

Storage Conditions

2 years -80 in solvent

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