ML221
Product Specifications
CAS Number
877636-42-5
Target
Angiotensin Receptor
Applications
GPCR & G Protein
Smiles
C1=CN=C (N=C1) SCC2=CC (=O) C (=CO2) OC (=O) C3=CC=C (C=C3) [N+] (=O) [O-]
Molecular Formula
C17H11N3O6S
Additionnal Information
ML221 is a potent apelin receptor (APJ) functional antagonist in cell-based assays that is >37-fold selective over the closely related angiotensin II type 1 (AT1) receptor. The IC50 values of ML221 are 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
VK472014-01 50 µg
Anti-HPV B19 NS1/Non-structural protein 1 Polyclonal Antibody
Sign In for Pricing
View Details VK472014-02 100 µg
Anti-HPV B19 NS1/Non-structural protein 1 Polyclonal Antibody
Sign In for Pricing
View Details MBS2133585-01 0.1 mL
Biotin Linked Monoclonal Antibody to Alpha1Antitrypsin (a1AT)
Sign In for Pricing
View Details MBS2133585-02 0.2 mL
Biotin Linked Monoclonal Antibody to Alpha1Antitrypsin (a1AT)
Sign In for Pricing
View Details MBS2133585-03 0.5 mL
Biotin Linked Monoclonal Antibody to Alpha1Antitrypsin (a1AT)
Sign In for Pricing
View Details