Derazantinib
Product Specifications
CAS Number
1234356-69-4
Synonyms
ARQ-087
Target
FGFR
Applications
Protein Tyrosine Kinase
Smiles
COCCNCCC1=CC (=CC=C1) NC2=NC=C3CC (C4=CC=CC=C4C3=N2) C5=CC=CC=C5F
Molecular Formula
C29H29FN4O
Additionnal Information
Derazantinib is an orally bioavailable inhibitor of the fibroblast growth factor receptor (FGFR) with IC50 values of 1.8 nM for FGFR2, and 4.5 nM for FGFR1 and 3, showing lower potency for FGFR4 (IC50=34 nM) . It also inhibits RET, DDR2, PDGFRβ, VEGFR and KIT.
Storage Conditions
3 years -20°C powder
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