Serabelisib (TAK-117)
Product Specifications
CAS Number
1268454-23-4
Synonyms
INK-1117, MLN-1117
Target
PI3K
Applications
PI3K/Akt/mTOR
Smiles
C1COCCN1C (=O) C2=CN=C3N2C=C (C=C3) C4=CC5=C (C=C4) OC (=N5) N
Molecular Formula
C19H17N5O3
Additionnal Information
Serabelisib (TAK-117, INK-1117, MLN-1117) is a potent and selective oral PI3Kα isoform inhibitor (IC50 of 21 nmol/L against PI3Kα) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kβ/γ/δ) and mTOR, and a high degree of selectivity against many other kinase.
Storage Conditions
2 years -80 in solvent
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