What is the catalog number for ARV-771?

The catalog number for ARV-771 is C13474-100mg.

What sizes are available for ARV-771?

ARV-771 is available in the following size(s): 100 mg.

ARV-771 is currently made to order / not held in immediate stock. Contact us for lead time.

ARV-771

Product Specifications

CAS Number

1949837-12-0

Target

PROTAC

Applications

Others

Smiles

CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NCCOCCCOCC (=O) NC (C (=O) N4CC (CC4C (=O) NC (C) C5=CC=C (C=C5) C6=C (N=CS6) C) O) C (C) (C) C) C7=CC=C (C=C7) Cl) C

Molecular Formula

C49H60ClN9O7S2

Additionnal Information

ARV-771 is a potent pan- (bromodomain and extra-terminal) BET degrader, a novel BET-PROTAC (proteolysis-targeting chimera) with Kd of 34 nM, 4.7 nM, 8.3 nM, 7.6 nM, 9.6 nM, and 7.6 nM for BRD2 (1), BRD2 (2), BRD3 (1), BRD3 (2), BRD4 (1), and BRD4 (2), respectively.