GSK180736A (GSK180736)
Product Specifications
CAS Number
817194-38-0
Target
GRK
Applications
GPCR & G Protein
Smiles
CC1=C (C (NC (=O) N1) C2=CC=C (C=C2) F) C (=O) NC3=CC4=C (C=C3) NN=C4
Molecular Formula
C19H16FN5O2
Additionnal Information
GSK180736A (GSK180736), developed as a Rho-associated, coiled-coil-containing protein kinase inhibitor, binds to GRK2 (G protein-coupled receptor kinase 2) with logIC50 pf -6.6 (logIC50 -4.0 for GRK5 and >-3 for GRK1) ; ≥400-fold selective for GRK2 over both GRK1 and GRK5.
Storage Conditions
2 years -80 in solvent
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