KG-501
Product Specifications
CAS Number
18228-17-6
Synonyms
2-naphthol-AS-E-phosphate
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
C1=CC=C2C=C (C (=CC2=C1) C (=O) NC3=CC=C (C=C3) Cl) OP (=O) (O) O
Molecular Formula
C17H13ClNO5P
Additionnal Information
KG-501 is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM) . It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay.
Storage Conditions
3 years -20°C powder
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