KG-501
Product Specifications
CAS Number
18228-17-6
Synonyms
2-naphthol-AS-E-phosphate
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
C1=CC=C2C=C (C (=CC2=C1) C (=O) NC3=CC=C (C=C3) Cl) OP (=O) (O) O
Molecular Formula
C17H13ClNO5P
Additionnal Information
KG-501 is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM) . It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay.
Storage Conditions
3 years -20°C powder
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
FAB2295S-100UG 100 µg
Human 4-1BB Ligand/TNFSF9 Alexa Fluor 750 Antibody
Sign In for Pricing
View Details MBS6211295-01 0.1 mL
EIF2S1 (Eukaryotic Translation Initiation Factor 2, Subunit 1 alpha, eIF2 alpha, eIF-2-alpha, eIF-2A, eIF-2alpha, EIF2A, Eukaryotic Translation Initiation Factor 2 Subunit 1) (MaxLight 550)
Sign In for Pricing
View Details MBS6211295-02 5x 0.1 mL
EIF2S1 (Eukaryotic Translation Initiation Factor 2, Subunit 1 alpha, eIF2 alpha, eIF-2-alpha, eIF-2A, eIF-2alpha, EIF2A, Eukaryotic Translation Initiation Factor 2 Subunit 1) (MaxLight 550)
Sign In for Pricing
View Details