GSK2193874
Product Specifications
CAS Number
1336960-13-4
Target
TRP Channel
Applications
Neuronal Signaling
Smiles
C1CCN (CC1) C2CCN (CC2) CC3=C (C4=C (C=C (C=C4) Br) N=C3C5=CC (=CC=C5) C (F) (F) F) C (=O) NC6 (CC6) C7=CC=CC=C7
Molecular Formula
C37H38BrF3N4O
Additionnal Information
GSK2193874 is an orally active, potent, and selective blocker of transient receptor potential vanilloid 4 (TRPV4) with IC50 values of 0.04 and 0.002 μM for hTRPV4 and rTRPV4, respectively.
Storage Conditions
2 years -80 in solvent
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