Lirametostat (CPI-1205)
Product Specifications
CAS Number
1621862-70-1
Synonyms
CPI 1205, CPI1205
Target
Histone Methyltransferase
Applications
Epigenetics
Smiles
CC1=CC (=C (C (=O) N1) CNC (=O) C2=C (N (C3=CC=CC=C32) C (C) C4CCN (CC4) CC (F) (F) F) C) OC
Molecular Formula
C27H33F3N4O3
Additionnal Information
Lirametostat (CPI-1205) is an orally available selective inhibitor of the histone lysine methyltransferase EZH2 with IC50 values of 2 nM and 52 nM for EZH2 and EZH1 respectively. It has potential antineoplastic activity.
Storage Conditions
2 years -80 in solvent
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