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PT2385

Product Specifications

CAS Number

1672665-49-4

Target

HIF

Applications

Angiogenesis

Smiles

CS (=O) (=O) C1=C2C (C (CC2=C (C=C1) OC3=CC (=CC (=C3) C#N) F) (F) F) O

Molecular Formula

C17H12F3NO4S

Additionnal Information

PT2385 is a HIF-2α antagonist with luciferase EC50 of 27 nM and no significant off-target activity.

Storage Conditions

3 years -20°C powder

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