CPI-637
Product Specifications
CAS Number
1884712-47-3
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1CC (=O) NC2=CC=CC (=C2N1) C3=CC4=C (C=C3) N (N=C4C5=CN (N=C5) C) C
Molecular Formula
C22H22N6O
Additionnal Information
CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor with IC50 values of 0.03 μM and 0.051μM for CBP and EP300 respectively in TR-FRET assay. It is highly selective against other bromodomains, displaying substantial biochemical activity only against BRD9.
Storage Conditions
2 years -80 in solvent
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